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Medicinal Chemistry
FACILE SYNTHESIS OF A 5-SULFAMOYLFURAN-2-CARBOXAMIDE LIBRARY. Gabriel Hum, Dana Razanno, Scott E. Collibee, Jason L. Davis
Program
Sunday
| Synthetic Organic | |||||||||||||||||
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1. |
ENZYMATIC RESOLUTION OF SUBSTITUTED MANDELIC ACIDS. John E. Reilly, Robert F. Campbell, Kevin Fitzpatrick, Larry Yet, Tord Inghardt, Olle Karlsson, Kristina Nilsson | ||||||||||||||||
| 2. | GENERATION OF 3-PYRIDYL BIARYL SYSTEMS VIA PALLADIUM-CATALYZED SUZUKI CROSS-COUPLING OF ARYL HALIDES WITH 3-PYRIDYLBOROXIN. Christopher L. Cioffi, William T. Spencer, Justin J. Richards, R. Jason Herr | ||||||||||||||||
| 3. | PALLADIUM-CATALYZED COUPLING OF ARYL IODIDES WITH ARYL BORONIC ACIDS. Jalal Haddad, Paul R. Bruzinski, Karen J. Jenkins, Daniel K. Keefe, Matthew Schiesher, Elisabeth Brot | ||||||||||||||||
| 4. | COMPUTATIONAL MODELS TO PREDICT BLOOD-BRAIN BARRIER PERMEATION AND CNS ACTIVITY. Douglas B. Kitchen, Govindan Subramanian | ||||||||||||||||
| 5. | MEDIAN PARTITIONING FOR COMPOUND SELECTION AND VIRTUAL SCREENING. John R. Furr, Douglas B. Kitchen, Jeffrey W. Godden, Jürgen Bajorath | ||||||||||||||||
| 6. | AN IMPROVED SYNTHESIS FOR THE LARGE SCALE PREPARATION OF SCHÖLLKOPF´S BIS-LACTIM ETHER CHIRAL AUXILIARIES. Nicholas J. Holman, Scott P. Corbin, Jianxie Chen | ||||||||||||||||
| 7. | A CONVENIENT GENERAL SYNTHETIC ROUTE TO BIARYL N-SUBSTITUTED IMIDAZOLES. Margaret B. Strickland, Pedro E. Hernández-Abad, Kejiang Hu, Carl Lindmark, Todd Luttrell, Jerod Robertson, Robert J. Duguid, Christopher Verbicky | ||||||||||||||||
| 8. | A GENERAL PROCEDURE FOR THE SYNTHESIS OF 2-SUBSTITUTED PYRIMIDINE-5-CARBOXYLIC ESTERS. David J. Fairfax, Paul Zhichkin, Shane A. Eisenbeis | ||||||||||||||||
| 9. | A PRACTICAL PROCESS FOR THE PREPARATION OF TRIMETHYLHYDRAZINE (TMH) AND ITS COUPLING WITH AN ACTIVATED ACID INTERMEDIATE. Silvina García Rubio, Deborah A. Renner, Chandra D. Wilson, John O. Rosser, Debasis Patra, Lawrence B. Fertel, J. Gregory Reid, Seemon H. Pines | ||||||||||||||||
| 10. | OXIDATIVE DEGRADATION OF VELCADE. Elisabeth Brot, Brian P. Haney, Kevin Hu, Chris Chiavelli, I. Fraser Pickersgill, John Bishop, Ian Parsons, Qing Lu, Ron Huang | ||||||||||||||||
| 11. | A MILD AND GENERAL METHOD FOR THE PREPARATION OF FUNCTIONALIZED ACYL HYDRAZONES. Chi-Hsin R. King, Paola Ciapetti, Moriyina D.C.E. Cole, Lori E. Awadalla, Charles R. Heap | ||||||||||||||||
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Medicinal Chemistry |
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| 12. | DESIGN AND SYNTHESIS OF PEPTIDE MIMETICS AS POTENTIAL INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 (PAI-1). Peter R. Guzzo, Michael P. Trova, George Lin, Tord Inghardt, Marcel Linschoten | ||||||||||||||||
| 13. | A STEREOSELECTIVE SYNTHESIS OF 24(S)-HYDROXYVITAMIN D2, A PRODRUG FOR 1-ALPHA-24(S)-DIHYDROXYVITAMIN D2. Chi-Hsin R. King, Lisa D. Coutts, William B. Geiss, Brian T. Gregg, Mark A. Helle, Mary E. Mateo, Zinovy Itov, Harold Meckler, Mark W. Zettler, Joyce C. Knutson | ||||||||||||||||
| 14. | 2-DIMETHYLAMINO-5-PHENYL-1,2,3,4-TETRAHYDRONA-PHTHALENES: A NEW CLASS OF LIGANDS FOR HISTAMINE H1 AND SEROTONIN 5HT2-TYPE RECEPTORS. Jacqueline A. Legere, Raymond G. Booth, Nader H. Moniri | ||||||||||||||||
| 15. | SYNTHESIS OF ENANTIOMERICALLY PURE (+)- AND (-)-18-METHOXYCORONARIDINE HYDROCHLORIDE AND THEIR PRELIMINARY ASSESSMENT AS ANTI-ADDICTIVE AGENTS. Chi-Hsin R. King, Harold Meckler, R. Jason Herr, Michael P. Trova, Stanley D. Glick, Isabelle M. Maisonneuve | ||||||||||||||||
| 16. | PREPARATION OF OPTICALLY ACTIVE (ACYLOXY)ALKYL ESTERS FROM OPTICALLY ACTIVE O-ACYL-ALPHA-HYDROXY ACIDS. Sean R. Dinn, Peter R. Guzzo, Jianhui Lu, Stefanie Oettinger-Loomis | ||||||||||||||||
| 17. | SYNTHESES OF CARBOXAMIDO-CONTAINING OPIATES VIA N-HYDROXY-SUCCINIMIDO ACTIVATED ESTERS. Mark P. Wentland, Rongliang Lou, Melissa A. VanAlstine, Xufeng Sun, Qun Lu, Yigong Bu, Jean M. Bidlack | ||||||||||||||||
| Parallel Synthesis | |||||||||||||||||
| 18. |
FACILE SYNTHESIS OF A 5-SULFAMOYLFURAN-2-CARBOXAMIDE LIBRARY. Gabriel Hum, Dana Razanno, Scott E. Collibee, Jason L. Davis |
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| 19. | MICROWAVE-ASSISTED SYNTHESIS OF 4-AMINOQUINAZOLINE DERIVATIVES VIA REACTION OF (2-CYANOPHENYL)-N,N-DIMETHYL FORMAMIDINES AND AMINES. David S. Yoon, Ying Han, Todd M. Stark, Sara B. Ruback, James C. Haber, Brian T. Gregg | ||||||||||||||||
| 20. | PARALLEL SYNTHESIS OF FUNCTIONAL FORMAMIDINES. Ying Han, Jennifer L. Butcher, Sara Ruback, Todd M. Stark, James C. Haber, David Yoon, Brian T. Gregg | ||||||||||||||||
| 21. | PARALLEL SYNTHESIS OF ETHYL QUINAZOLINE-2-CARBOXYLATE DERIVATIVES. James C. Haber, Ying Han, Dmytro Tymoshenko, M. Todd Luttrell | ||||||||||||||||
| NANOTECHNOLOGY | |||||||||||||||||
| 22. | PHOTOACTIVATED LUMINESCENCE OF CADMIUM SELENIDE QUANTUM DOTS. Zhouying Zhao, G. Sirinakis, A. Tayi, Michael A. Carpenter | ||||||||||||||||
| 23. | TAILORED NANOMATERIALS: HIGHLY SELECTIVE & SENSITIVE CHEMICAL SENSORS FOR HYDROCARBON ANALYSIS. George Sirinakis, Z. Zhao, Y. Sevryugina, M. Petrukhina, Michael A. Carpenter, A. Tayi | ||||||||||||||||
| ORIGINS OF LIFE | |||||||||||||||||
| 24. | THE ORIGINS OF LIFE AND INTERCALATOR-MIEDIATED LIGATION OF NUCLEIC ACIDS WITH BASES. Brooke Rosenzweig | ||||||||||||||||
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Program |
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