36th Middle Atlantic Regional Meeting (MARM)
June 8-11   2003
Spnsored by the Trenton ACS Section and
Princeton University


Confirmed Speakers: General Medicinal Chemistry


Chair: Dr. T. Caggiano Wyeth Pharmaceuticals

Sponsored by:






Program Id Author Name Author Institution Title Presentation Time Building Room
12 Paul Anderson Independent Consultant EVOLUTION OF MODERN DRUG DISCOVERY Monday, Jun 9 2003 9:00AM Jadwin JA10
13 Frank Koehn Wyeth Research RAISING THE IMPACT OF NATURAL PRODUCTS IN MODERN DRUG DISCOVERY Monday, Jun 9 2003 9:40AM Jadwin JA10
14 Edmund Graziani Wyeth Research NATURAL PRODUCTS CHEMISTRY AT WYETH RESEARCH: RECENT PROGRESS IN GENERATING LEADS FOR DRUG DISCOVERY Monday, Jun 9 2003 10:00AM Jadwin JA10
15 John W. Clader PH.D. Pharmaceutical FROM SERENDIPITY TO DESIGN: THE DISCOVERY OF EZETIMIBE AND OTHER NOVEL CHOLESTEROL ABSORPTION INHIBITORS Monday, Jun 9 2003 10:20AM Jadwin JA10
16 Thomas Edward D'Ambra Albany Molecular Research, Inc. SHORT HISTORY AND IMPACT OF CHEMISTRY OUTSOURCING COMPANIES ON DRUG DISCOVERY AND DEVELOPMENT. A SUPPLIERS VIEW Monday, Jun 9 2003 11:00AM Jadwin JA10
17 Robert Hormann RHeoGene, LLC MULTIDIMENSIONAL QSAR AND SUPERIMPOSITION EVALUATION OF ECDYSONE RECEPTOR GENE-SWITCH ACTUATORS Monday, Jun 9 2003 11:40AM Jadwin JA10
PM Session
Program Id Author 1 Name Author 1 Institution Title Presentation Time Building Room
73 S. David Kimball Lexicon Pharmaceuticals CHALLENGES IN DRUG DISCOVERY IN THE 21ST CENTURY: TARGET VALIDATION Monday, Jun 9 2003 2:30PM Jadwin JA10
74 Timothy A. Blizzard Merck Research Labs 2-PHENYLSPIROINDENES AND 2-PHENYLSPIROINDENEDIONES AS NOVEL ESTROGEN RECEPTOR LIGANDS Monday, Jun 9 2003 3:10PM Jadwin JA10
75 Bart L. DeCorte Johnson & Johnson Pharmaceutical Research & Development DISCOVERY OF TMC125, A NEXT GENERATION NNRTI WITH ACTIVITY AGAINST SINGLE AND DOUBLE MUTANTS Monday, Jun 9 2003 3:30PM Jadwin JA10
76 Robert Aslanian Schering-Plough Research Institute DISCOVERY OF SCH 79687, A NOVEL IMIDAZOLE-BASED ANTAGONIST OF THE H3 RECEPTOR Monday, Jun 9 2003 4:00PM Jadwin JA10
77 Louis Lombardo Bristol-Myers Squibb Pharmaceutical Research Institute STUDIES DIRECTED TOWARDS THE IDENTIFICATION OF SMALL-MOLECULE INHIBITORS OF FARNESYL PROTEIN TRANSFERASE FOR ONCOLOGY INDICATIONS Monday, Jun 9 2003 4:35PM Jadwin JA10
78 Regine S Bohacek Boston DeNovo AlleGrow and FLO+: New Tools for Drug Design Monday, Jun 9 2003 5:10PM Jadwin JA10
Last modified: Mon May 26 15:16:25 2002